BX-912
- SMILES: Brc1cnc(Nc2cccc(NC(=O)N3CCCC3)c2)nc1NCCc1c[nH]cn1
- Formula: C20H23BrN8O
- Purity: 0.9934
- CAS#: 702674-56-4
- Molecular Weight: 471.363
- Bioactivity: BX-912 is a specific inhibitor of 3-Phosphoinositide-dependent Kinase-1 (PDK1, IC50: 12 nM). The selectivity of BX-912 is more 10 fold than C-Kit, EGFR, PKA, PKC etc.
For research use only.
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