ARP-100

ARP-100

• SMILES: O=C(NO)CN(OC(C)C)S(=O)(=O)C=1C=CC(=CC1)C=2C=CC=CC2
• Formula: C17H20N2O5S

• Purity: 0.9834
• CAS#: 704888-90-4
• Molecular Weight: 364.42
• Bioactivity: ARP-100 is a potent and selective matrix metalloproteinase MMP-2 inhibitor (IC50=12 nM). ARP-100 interacts with the S1' pocket of MMP-2 and exhibits anti-invasive properties in an in vitro invasion Matrigel model. ARP-100 has low inhibitory activity against MMP-1 (>50 μM), MMP-3 (4.5 μM), MMP-7 (>50 μM) and MMP-9 (0.2 μM)[1][2].

For research use only.